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Compound 101

Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3.

Product Specifications

CAS Number

865608-11-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

466.468

Molecular Formula

C24H21F3N6O

Notes

Research use only, not for human use.

Receptor

GRK (GPCRK)

Available Sizes

Curated Selection

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