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CDK5 inhibitor 20-223

CDK5 inhibitor 20-223 (CP 668863) potent, selective, ATP-competitive CDK2/5 inhibitor with IC50 of 6.0 and 8.8 nM for CDK2/CyclinE and CDK5/p35, with little to no activity against CDK1/4/6/7/9.

Product Specifications

CAS Number

865317-30-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

305.381

Molecular Formula

C19H19N3O

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Curated Selection

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