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GSK598809

GSK598809 (GSK-598809) is a potent, selective, CNS penetrant and orally bioavailable dopamine D3 receptor antagonist with pKi of 8.9; displays >100-fold selectivity over D2 and H1 receptors.

Product Specifications

CAS Number

863680-45-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

481.514

Molecular Formula

C22H23F4N5OS

Notes

Research use only, not for human use.

Receptor

Dopamine Receptor

Available Sizes

Curated Selection

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