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LY2228820 dimesylate

LY2228820 dimesylate (Ralimetinib) is a potent, selective, orally available inhibitor p38 MAPK with IC50 of 5.3 and 3.2 nM for p38α and p38β, respectively.

Product Specifications

CAS Number

862507-23-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

612.737

Molecular Formula

C26H37FN6O6S2

Notes

Research use only, not for human use.

Receptor

P38α

Available Sizes

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