Sapitinib
Sapitinib (AZD-8931, AZD8931) is a equipotent, reversible inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4. 3 and 4 nM (phosphorylation inhibition), respectively.
Product Specifications
CAS Number
848942-61-0
Stability
≥ 2 years
Purity
>98% (HPLC)
Weight
473.9277
Molecular Formula
C23H25ClFN5O3
Notes
Research use only, not for human use.
Receptor
EGFR|HER2/ErbB2
Available Sizes
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