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Sapitinib

Sapitinib (AZD-8931, AZD8931) is a equipotent, reversible inhibitor of EGFR, ErbB2 and ErbB3 with IC50 of 4. 3 and 4 nM (phosphorylation inhibition), respectively.

Product Specifications

CAS Number

848942-61-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

473.9277

Molecular Formula

C23H25ClFN5O3

Notes

Research use only, not for human use.

Receptor

EGFR|HER2/ErbB2

Available Sizes

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