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Bitopertin

A potent and selective GlyT1 inhibitor with EC50 of 30 nM; no activity for GlyT2, hERG, CYP450 enzymes above 10 uM.

Product Specifications

CAS Number

845614-11-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

543.455

Molecular Formula

C21H20F7N3O4S

Notes

Research use only, not for human use.

Receptor

GlyT1

Available Sizes

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