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GSK983

GSK983 (GSK-983) is a potent, cell penetrant PCAF/GCN5 PROTAC, induces concentration-dependent degradation of PCAF and GCN5 in THP1 cells with DC50 value of 1.5 nM and 3 nM, respectively.

Product Specifications

CAS Number

827591-02-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

895.856

Molecular Formula

C45H51BrN8O7

Notes

Research use only, not for human use.

Receptor

PROTAC

Available Sizes

Curated Selection

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