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Palbociclib hydrochloride

A potent and selective inhibitor of CDK4/6 with IC50 of 11 nM/16 nM; no inhibition for CDK2A (IC50>5 uM) ; inhibits MDA-MB453 cells with IC50 of 0.16 uM.

Product Specifications

CAS Number

827022-32-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

483.9937

Molecular Formula

C24H30ClN7O2

Notes

Research use only, not for human use.

Receptor

CDK2/CyclinA|CDK2/CyclinE2|CDK4/CyclinD1|CDK4/CyclinD3|CDK6/CyclinD2

Available Sizes

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