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Rislenemdaz hydrochloride

Rislenemdaz (MK 0657; CERC 301) is a potent, orally bioavailable, brain‐penetrant, NR2B-selective NMDA receptor (GluN2B) antagonist with Ki and IC 50 of 8.1 nM and 3.6 nM respectively.

Product Specifications

CAS Number

808733-06-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

394.875

Molecular Formula

C19H24ClFN4O2

Notes

Research use only, not for human use.

Receptor

IGluR

Available Sizes

Curated Selection

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