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XL-647

XL-647 (Tesevatinib, EXEL-7647, KD-019) is a novel spectrum-selective kinase inhibitor that potently inhibits the EGFR, ErbB2, KDR and EphB4 with IC50 of 0.3, 16, 1.5 and 1.4 nM, respectively.

Product Specifications

CAS Number

781613-23-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

491.4

Molecular Formula

C24H25Cl2FN4O2

Notes

Research use only, not for human use.

Receptor

EGFR

Available Sizes

Curated Selection

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