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GNF-5

GNF-5, an analogue of GNF-2 with improved pharmacokinetic properties, is a selective non-ATP competitive inhibitor of Bcr-Abl with an IC50 value of 0.22±0.1 uM (Wild type Abl) .

Product Specifications

CAS Number

778277-15-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

418.37

Molecular Formula

C20H17F3N4O3

Notes

Research use only, not for human use.

Receptor

Bcr-Abl

Available Sizes

Frequently Asked Questions

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