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TAE226

NVP-TAE226 is a potent FAK inhibitor with IC50 of 5.5 nM and modestly potent to Pyk2 (IC50=3.5 nM) ; 10- to 100-fold less potent against InsR, IGF-1R, ALK, and c-Met.

Product Specifications

CAS Number

761437-28-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

468.94

Molecular Formula

C23H25ClN6O3

Notes

Research use only, not for human use.

Receptor

C-Met| FAK| IGF-1R| Insulin Receptor| PYK2

Available Sizes

Curated Selection

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