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K-777

K-777 is a potent and selective CCR4 antagonist that inhibits both CCL17 binding and CCL17-induced chemotaxis in Hut78 cells with IC50 of 57 and 8.9 nM respectively.

Product Specifications

CAS Number

749860-43-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

641.5

Molecular Formula

C28H32F4IN5

Notes

Research use only, not for human use.

Receptor

Chemokine Receptor

Available Sizes

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