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Neratinib

A potent, highly selective, irreversible HER2 and EGFR inhibitor with IC50 of 59 nM and 92 nM in cell-free assays.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

557.0427

Molecular Formula

C30H29ClN6O3

Notes

Research use only, not for human use.

Receptor

EGFR|HER2|PDK1|Src|VEGFR2 (KDR)

CAS Number

698387-09-6

Available Sizes

Curated Selection

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