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BRD6989

A novel potent, selective CDK8 inhibitor with IC50 of 0.5 uM against recombinant Cyclin C/CDK8 complex; displays no activity against several CDKs involved in cell cycle including CDK19 (IC50>30 uM) .

Product Specifications

CAS Number

642008-81-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

264.332

Molecular Formula

C16H16N4

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Curated Selection

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