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ARC 239 dihydrochloride

A potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.

Product Specifications

CAS Number

55974-42-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

480.43

Molecular Formula

C24H29N3O3.2HCl

Notes

Research use only, not for human use.

Receptor

Adrenergic Receptor

Available Sizes

Curated Selection

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