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UC-857993

A small molecule inhibitor of guanine nucleotide exchange factor (GEF) catalytic activity that binds to SOS1 (Kd=14.7 uM) and disrupts GEF-Ras interaction.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

403.906

Molecular Formula

C25H22ClNO2

Notes

Research use only, not for human use.

Receptor

Ras

CAS Number

487001-04-7

Available Sizes

Curated Selection

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