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Pitolisant oxalate

A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM; no effect on H1, H2, H4 receptors (IC50>10 uM) .

Product Specifications

CAS Number

362665-57-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

385.8823

Molecular Formula

C19H28ClNO5

Notes

Research use only, not for human use.

Receptor

Histamine Receptor

Available Sizes

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