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AZD-9056 hydrochloride

A potent, selective, orally bioavailable P2X7 receptor antagonist; inhibits release of pro-inflammatory mediators from isolated human peripheral monocytes (IL-1β and IL-18) and human alveolar macrophages (IL-1β) with IC50 values of 10-13 nM.

Product Specifications

CAS Number

345303-91-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

455.46084

Molecular Formula

C24H36Cl2N2O2

Notes

Research use only, not for human use.

Receptor

P2X Receptor

Available Sizes

Curated Selection

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