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MRK-016

A potent, functionally selective, CNS-penetrating and orally bioavailable inverse agonist of benzodiazepine site of GABAA α5 receptor.

Product Specifications

CAS Number

342652-67-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

368.3931

Molecular Formula

C17H20N8O2

Notes

Research use only, not for human use.

Receptor

GAT

Available Sizes

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