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NPS-2143 hydrochloride

A potent, selective and orally active CaSR antagonist with IC50 of 43 nM; does not inhibit cytoplasmic Ca2+ responses to glutamate in HEK 293 cells engineered to express mGluRs and GABAB receptors.

Product Specifications

CAS Number

324523-20-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

445.3814

Molecular Formula

C24H26Cl2N2O2

Notes

Research use only, not for human use.

Receptor

CaSR

Available Sizes

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