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VX-765

VX-765 (Belnacasan) is an orally absorbed prodrug of VRT-043198, which is a potent and selective inhibitor of interleukin-converting enzyme/caspase-1 with Ki of 0.8 nM.

Product Specifications

CAS Number

273404-37-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

508.995

Molecular Formula

C24H33ClN4O6

Notes

Research use only, not for human use.

Receptor

Caspase-1|Caspase-4

Available Sizes

Frequently Asked Questions

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