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TPA023

TPA023 is a potent, α2/α3 subtype-selective, and oral GABAA receptor agonist with Kd of 0.92, 1.05 and 0.58 nM for α1-, α2-, α3-, and α5-containing human receptors.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

395.442

Molecular Formula

C20H22FN7O

Notes

Research use only, not for human use.

Receptor

GAT

CAS Number

252977-51-8

Available Sizes

Curated Selection

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