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HSD992

HSD992 is a potent, selective CDK2/3 inhibitor with moderate CDK9 inhibition with IC50 of 18 nM, 57 nM and 49 nM for CDK3/cyclin E, CDK2/cyclin A1 and CDK2/cyclin E, respecively.

Product Specifications

CAS Number

2222045-50-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

370.474

Molecular Formula

C22H18N4S

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Curated Selection

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