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GW-8510

GW-8510 (GW8510) is a potent, selective inhibitor of CDK2 with IC50 of 10 nM; displays weak inhibition for CDK1 and CDK4 (IC50=110 and 130 nM, respectively) in vitro biochemical assays.

Product Specifications

CAS Number

222036-17-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

449.51

Molecular Formula

C21H15N5O3S2

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Frequently Asked Questions

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