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PD-184352

A potent, ATP non-competitive MEK1/2 inhibitor with IC50 of 17 nM in cell-based assays, displays 100-fold more selective for MEK1/2 than MEK5.

Product Specifications

CAS Number

212631-79-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

478.6595

Molecular Formula

C17H14ClF2IN2O2

Notes

Research use only, not for human use.

Receptor

MEK1|MEK2

Available Sizes

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