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WHI-P154

WHI-P154 is a potent JAK3 inhibitor with IC50 of 1.8 μM, no activity against JAK1 or JAK2, also inhibits EGFR, Src, Abl, VEGFR and MAPK, prevents Stat3, but not Stat5 phosphorylation.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

376.2

Molecular Formula

C16H14BrN3O3

Notes

Research use only, not for human use.

Receptor

EGFR| JAK3| Src| VEGFR

CAS Number

211555-04-3

Available Sizes

Curated Selection

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