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LOXO-195

LOXO-195 (Selitrectinib; LOXO 195, LOXO195) is a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively.

Product Specifications

CAS Number

2097002-61-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

380.427

Molecular Formula

C20H21FN6O

Notes

Research use only, not for human use.

Receptor

Trk Receptor

Available Sizes

Curated Selection

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