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OTX015

OTX015 is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4. Phase 1.

Product Specifications

CAS Number

202590-98-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

491.99

Molecular Formula

C25H22ClN5O2S

Notes

Research use only, not for human use.

Receptor

BRDs

Available Sizes

Frequently Asked Questions

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