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CDK inhibitor E9

CDK inhibitor E9 is a novel CDK inhibitor that can overcomes ABC-mediated resistance of THZ1, functions as a potent, non-covalent inhibitor of CDK9 and a covalent inhibitor of CDK12.

Product Specifications

CAS Number

2020052-55-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

434.544

Molecular Formula

C24H30N6O2

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

Curated Selection

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