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MMSET-IN-1

MMSET-IN-1 is a potent, selective epigenetic oncogene MMSET (aka NSD2 or WHSC1) inhibitor with Ki/IC50 of 1.6/3.3 uM.

Product Specifications

CAS Number

1998139-29-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

423.474

Molecular Formula

C18H29N7O5

Notes

Research use only, not for human use.

Receptor

HMTase

Available Sizes

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