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GNE-272

A potent and selective the bromodomains of CBP/EP300 inhibitor with IC50 of 0.02 and 0.03 uM for CBP and EP300, respectively.

Product Specifications

CAS Number

1936428-93-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

424.48

Molecular Formula

C22H25FN6O2

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

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