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GNE-049

GNE-049 (GNE049) is a potent, selective, orally available inhibitor of CBP/p300 bromodomain with biochemical IC50 of 1.1/2.3 nM, respectively.

Product Specifications

CAS Number

1936421-41-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

510.59

Molecular Formula

C27H32F2N6O2

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

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