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LY3295668

LY3295668 (LY-3295668, AK-01) is a novel potent, highly selective, orally active Aurora-A kinase inhibitor with Ki of 0.8 nM, H446 AurA auto-P IC50 of 0.6 nM.

Product Specifications

CAS Number

1919888-06-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

489.952

Molecular Formula

C24H26ClF2N5O2

Notes

Research use only, not for human use.

Receptor

Aurora Kinase

Available Sizes

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