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GLPG-2222

GLPG-2222 (ABBV-2222, Galicaftor) is a novel potent and efficacious CFTR corrector with EC50 of 5 nM; is highly potent (5 nM) and efficacious in cells from multiple CF patient donors that have F508del homozygous mutation.

Product Specifications

CAS Number

1918143-53-9

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

559.47

Molecular Formula

C28H21F4NO7

Notes

Research use only, not for human use.

Receptor

CFTR

Available Sizes

Frequently Asked Questions

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