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GSK-6853

A potent, highly selective and cell-active BRPF1 bromodomain inhibitor with TR-FRET pIC50 of 8.1.

Product Specifications

CAS Number

1910124-24-1

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

409.4815

Molecular Formula

C22H27N5O3

Notes

Research use only, not for human use.

Receptor

BRPF1|BRPF2|BRPF3

Available Sizes

Curated Selection

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