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CPI-637

A potent and selective, cell-active CBP/EP300 bromodomain inhibitor with CBP BRET EC50 of 0.03 uM.

Product Specifications

CAS Number

1884712-47-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

386.4497

Molecular Formula

C22H22N6O

Notes

Research use only, not for human use.

Receptor

BRD4|CBP|EP300

Available Sizes

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