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EFT508

EFT508 (Tomivosertib) is a potent, highly selective, reversible, ATP-competitive, and orally bioavailable MNK1 and MNK2 inhibitor with IC50 of 1-2 nM in enzyme assays.

Product Specifications

CAS Number

1849590-01-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

340.3797

Molecular Formula

C17H20N6O2

Notes

Research use only, not for human use.

Receptor

MNK1|MNK2

Available Sizes

Curated Selection

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