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Gefitinib

A potent, selective, orally active EGFR inhibitor with IC50 of 23 nM; inhibits EGF-stimulated proliferation of KB cells with IC50 of 80 nM.

Product Specifications

CAS Number

184475-35-2

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

446.9024

Molecular Formula

C22H24ClFN4O3

Notes

Research use only, not for human use.

Receptor

Tyr1173 (NR6W cells) | Tyr1173 (NR6wtEGFR cells) | Tyr992 (NR6W cells) | Tyr992 (NR6wtEGFR cells)

Available Sizes

Curated Selection

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