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ARV-825

ARV-825 is a hetero-bifunctional PROTAC (Proteolysis Targeting Chimera) that recruits BRD4 to the E3 ubiquitin ligase cereblon, leading to fast, efficient, and prolonged degradation of BRD4 via the proteasome.

Product Specifications

CAS Number

1818885-28-7

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

923.4316

Molecular Formula

C46H47ClN8O9S

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

Curated Selection

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