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ARV-825

ARV-825 is a hetero-bifunctional PROTAC (Proteolysis Targeting Chimera) that recruits BRD4 to the E3 ubiquitin ligase cereblon, leading to fast, efficient, and prolonged degradation of BRD4 via the proteasome.

Product Specifications

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

923.4316

Molecular Formula

C46H47ClN8O9S

Notes

Research use only, not for human use.

Receptor

Bromodomain

CAS Number

1818885-28-7

Available Sizes

Curated Selection

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