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THIQ 40

THIQ 40 (THIQ40) is a potent, orally available ERα antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERα binding) and 30 nM (ERα transcription), IC50 of 0.9 nM (ERα degradation) .

Product Specifications

CAS Number

1799430-91-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

427.544

Molecular Formula

C28H29NO3

Notes

Research use only, not for human use.

Receptor

Estrogen Receptor/ERR

Available Sizes

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