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Nepicastat hydrochloride

Nepicastat (RS-25560-197, SYN-117) is a potent, selective, orally active inhibitor of dopamine-beta-hydroxylase (DBH) with IC50 of 8.5 and 9.0 nM for bovine and human DBH, respectively.

Product Specifications

CAS Number

170151-24-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

331.8

Molecular Formula

C14H16ClF2N3S

Notes

Research use only, not for human use.

Receptor

Dopamineβ-hydroxylase

Available Sizes

Curated Selection

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