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BI 894999

BI 894999 is a novel potent, selective BET inhibitor with IC50 of 5 and 41 nM for BRD4-BD1 and BRD4-BD2 bromodomains, respectively.

Product Specifications

CAS Number

1660117-38-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

429.524

Molecular Formula

C25H27N5O2

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

Curated Selection

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