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Naltrexone

A potent, competitive antagonist for μ, κ, δ, and σ-opioid receptors with Ki of 0.0825 nM, 0.509 nM, and 8.02 nM, for MOR, KOR, and DOR, respectively.

Product Specifications

CAS Number

16590-41-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

341.4009

Molecular Formula

C20H23NO4

Notes

Research use only, not for human use.

Receptor

Opioid Receptor

Available Sizes

Curated Selection

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