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GS-626510

GS-626510 (GS-6510, GS 6510, GS 626510) is a novel BET family bromodomains inhibitor with Kd of 0.5-2.8 nM for BRD2/3/4, and BRDT.

Product Specifications

CAS Number

1637770-13-8

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

394.478

Molecular Formula

C25H22N4O

Notes

Research use only, not for human use.

Receptor

Bromodomain

Available Sizes

Curated Selection

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