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KZR-616

KZR-616 (KZR616) is a potent, selective dual immunoproteasome subunit LMP7/LMP2 inhibitor with IC50 of 39 nM/139 nM, weakly inhibits β5, MECL-1 and no acitivty against β1 subunit.

Product Specifications

CAS Number

1629677-75-3

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

586.686

Molecular Formula

C30H42N4O8

Notes

Research use only, not for human use.

Receptor

Proteasome

Available Sizes

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