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GLPG-1690

GLPG-1690 (Ziritaxestat, GLPG1690) is a first-in-class, potent, competitive autotaxin inhibitor with Ki/IC50 of 15 nM/131 nM.

Product Specifications

CAS Number

1628260-79-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

588.71

Molecular Formula

C30H33FN8O2S

Notes

Research use only, not for human use.

Receptor

Autotaxin

Available Sizes

Frequently Asked Questions

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