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G1T38

G1T38 (Lerociclib, G1T 38) is a novel, potent and selective inhibitor of CDK4/6 with biochemical IC50 of 1 nM and 2 nM for CDK4/cyclin D1 and CDK6/cyclin D3, respectively.

Product Specifications

CAS Number

1628256-23-4

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

474.613

Molecular Formula

C26H34N8O

Notes

Research use only, not for human use.

Receptor

CDK

Available Sizes

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